APIM050131: CO-1686 (ROCILETINIB)
CAS No.: 1374640-70-6.
Purity: >99.5% (HPLC at 214 and 254 nm).
QC: HPLC-MS, 1HNMR and Quantitative Elemental Analysis.
Solubility: Soluble in DMSO.APIM050132: CRENOLANIB
CAS No.: 670220-88-9.
Purity: >99.5% (HPLC).
QC: HPLC-MS, 1HNMR, and Quantitative Elemental Analysis.
Solubility: Soluble in DMSO, and water with 1 eq. of acid.APIM050312: AG-221 (ENASIDENIB)
CAS No.: 1446502-11-9.
Purity: >99.5% by HPLC at 214 and 254 nm.
QC: HPLC-MS, 1H-NMR and Quantitative Elemental Analysis Report.
Solubility: Refer to Certificate.APIM050043: LY3381916
CAS No.: 2166616-75-5.
Purity: >99.5% by Achiral and Chiral HPLCs.
QC: Achiral and Chiral HPLCs, MS, 1H-NMRs, and Quantitative Elemental Analysis Report.
Solubility: Refer to Certification of Analysis.APIM050024: BMN-673 (Talazoparib) (MDV-3800)
CAS No.: 1207456-01-6.
Purity: 100% Optically Pure (Chiral HPLC), 99.3%-99.5% chemically Pure by Achiral HPLC at 214 and 254 nm.
QC: Achiral and Chiral HPLCs, NMR and Quantitative Elemental Analysis Report.
Solubility: Refer to Certificate of Analysis.APIM050294: AZD5582
CAS No.: 1258392-53-8.
Purity: ≥99% purity (HPLC).
QC: HPLC-MS, 1HNMR, and Quantitative Elemental Analysis.
Solubility: Soluble in DMSO, Water.APIM050051: MLN7243 (TAK-243, AOB 87172)
CAS No.: 1450833-55-2.
Purity: 100% Stereomerical Purity (Chiral HPLC), 99% Chemical Purity (HPLC at 220 and 254 nm),.
QC: HPLC-MS, 1HNMR, Chiral HPLC, and Quantitative Elemental Analysis.
Solubility: Soluble in DMSO.APIM050027: CB-1158 (INCB01158)
CAS No.: 2095732-06-0.
Purity: 99% by achiral and chiral HPLCs ( detected at 210 nm wavelength).
QC: Achiral and Chiral HPLCs, MS, NMR and Quantitative Elemental Analysis.
Solubility: >100mM in Water.APIM050006: ADU-S100 (MIW815)
CAS No.: 1638750-95-4 (Sodium Salt), 1638241-89-0 (Free Acid)
Purity: >99.5% by HPLC (at 214 nm).
QC: HPLC, MS, 1H-, 31P-NMRs,
Solubility: Water (>36.7mg/ml, >50 mM).APIM050078: AP26113 (BRIGATINIB)
CAS No.: 1197953-54-0.
Purity: >99% by HPLC.
QC: HPLC-MS, NMR and Quantitative Elemental Analysis.
Solubility: Soluble in DMSO.